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Covalent/irreversible inhibitors target the redox/catalytic apparatus of TGR with almost no recognition elements that give affinity and selectivity for TGR over off-targets and the cellular redox apparatus resulting in undesirable cross-reactions and low specificity in vivo 25

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10.3390/ijms25179715 148

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Ursodeoxycholate stimulates Na+-H+ exchange in rat liver basolateral plasma membrane vesicles

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J Physiol 465: 303323

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